SCHEMBL4540431

SCHEMBL4540431

O=C(CC1CCN(S(=O)(=O)c2ccccc2)C1)NC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
KMT2A Q03164 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
EPHX1 P07099 5/20 0.51
ALDH1A1 P00352 4/20 0.47
LMNA P02545 3/20 0.47
TSHR P16473 1/20 0.47
ALOX12 P18054 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4537427 0.95 SMN1; SMN2 (0.52) NPC1RAB9AKMT2ASMN1; SMN2EPHX1
SCHEMBL4543052 0.94 NPC1 (0.48) NPC1RAB9AKMT2ASMN1; SMN2EPHX1
SCHEMBL4542094 0.93 NPC1 (0.57) NPC1RAB9AKMT2ASMN1; SMN2EPHX1
SCHEMBL4539274 0.89 CYP3A4 (0.51) NPC1KMT2AEPHX1ALDH1A1LMNA
SCHEMBL4536776 0.89 LMNA (0.62) NPC1RAB9AKMT2ASMN1; SMN2EPHX1
SCHEMBL4535944 0.89 EPHX1 (0.52) RAB9AEPHX1ALDH1A1LMNATSHR
SCHEMBL4537257 0.88 LMNA (0.51) NPC1RAB9AKMT2ASMN1; SMN2EPHX1
SCHEMBL4539985 0.88 TSHR (0.50) NPC1RAB9AKMT2ASMN1; SMN2EPHX1
SCHEMBL4539809 0.88 HSD11B1 (0.52) NPC1RAB9AKMT2ASMN1; SMN2EPHX1
SCHEMBL8053303 0.88 HSD11B1 (0.52) NPC1RAB9AKMT2ASMN1; SMN2EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed