SCHEMBL4539274

SCHEMBL4539274

O=C(CC1CCN(S(=O)(=O)c2ccc(F)cc2)C1)NC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.51
CYP2C19 P33261 1/20 0.51
EPHX1 P07099 2/20 0.49
ALDH1A1 P00352 4/20 0.48
LMNA P02545 3/20 0.48
HTT P42858 2/20 0.48
TSHR P16473 1/20 0.48
ALOX12 P18054 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
MAPT P10636 1/20 0.46
PKM P14618 1/20 0.45
CCR3 P51677 1/20 0.45
KMT2A Q03164 2/20 0.44
EPHX2 P34913 2/20 0.43
NPC1 O15118 1/20 0.43
KDM4E B2RXH2 1/20 0.43
POLB P06746 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4530361 0.95 CYP3A4 (0.59) CYP3A4CYP2C19EPHX1ALDH1A1LMNA
SCHEMBL4536795 0.94 EPHX1 (0.54) EPHX1ALDH1A1LMNAHTTTSHR
SCHEMBL8069615 0.91 EPHX1 (0.47) CYP3A4CYP2C19EPHX1ALDH1A1LMNA
SCHEMBL4542516 0.90 LMNA (0.49) EPHX1ALDH1A1LMNAHTTTSHR
SCHEMBL4536776 0.89 LMNA (0.62) CYP3A4EPHX1ALDH1A1LMNAHTT
SCHEMBL4535944 0.89 EPHX1 (0.52) EPHX1ALDH1A1LMNAHTTTSHR
SCHEMBL4540431 0.89 NPC1 (0.55) EPHX1ALDH1A1LMNAHTTTSHR
SCHEMBL4539985 0.88 TSHR (0.50) EPHX1ALDH1A1LMNAHTTTSHR
SCHEMBL4543052 0.88 NPC1 (0.48) EPHX1ALDH1A1LMNAHTTTSHR
SCHEMBL4540032 0.87 PKM (0.51) EPHX1ALDH1A1LMNAHTTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed