SCHEMBL4540918

SCHEMBL4540918

COC(=O)CCc1ccc(N2CCNCC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 4/20 0.50
HTR3E A5X5Y0 2/20 0.50
HTR3B O95264 2/20 0.50
HTR3A P46098 2/20 0.50
HTR3D Q70Z44 2/20 0.50
HTR3C Q8WXA8 2/20 0.50
SIGMAR1 Q99720 2/20 0.50
MAPT P10636 2/20 0.47
MAPKAPK2 P49137 2/20 0.46
HRH3 Q9Y5N1 1/20 0.46
AOC3 Q16853 3/20 0.46
ALDH1A1 P00352 2/20 0.46
USP2 O75604 1/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
USP28 Q96RU2 4/20 0.45
USP25 Q9UHP3 3/20 0.45
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
IRAK4 Q9NWZ3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10899752 0.85 ALDH1A1 (0.57) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7312990 0.85 ADRB1 (0.43) ADRB1HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL7366386 0.84 ALDH1A1 (0.56) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2302994 0.82 ITGB3 (0.61) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL10899597 0.82 ME2 (0.55) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL29414364 0.82 ME2 (0.51) MAPTALDH1A1ITGB3ITGA2B
Hydrochloric Acid SCHEMBL7396017 0.81 DRD2 (0.46) HRH3ITGB3ITGA2B
SCHEMBL3684659 0.79 USP28 (0.48) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL3680077 0.79 NPC1 (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
Acetic Acid Methyl Ester SCHEMBL27846699 0.78 ADRB1 (0.51) ADRB1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064569-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-18 WO disclosed
US-5994356-A ANTICOAGULANT KARL THOMAE (DE) 1999-11-30 US disclosed
EP-0892783-A1 CARBOXYLIC ACID DERIVATIVES WITH AN AGGREGATION-INHIBITING ACTION Dr. Karl Thomae GmbH (DE) 1999-01-27 EP disclosed
WO-1997037975-A1 CARBOXYLIC ACID DERIVATIVES WITH AN AGGREGATION-INHIBITING ACTION DR. KARL THOMAE GMBH (DE) 1997-10-16 WO disclosed