SCHEMBL4544118

SCHEMBL4544118

COc1ccc2c(c1)c(C(=O)c1nnc(-c3ccccn3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl.Cc1ccc2c(c1)c(C(=O)c1nnc(-c3ccccn3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1.O=C(c1nnc(-c2ccccn2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccc(Cl)cc12.O=C(c1nnc(-c2ccccn2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 2/20 0.38
ACHE P22303 1/20 0.37
FAAH O00519 1/20 0.37
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
RGS12 O14924 1/20 0.35
CYP1A2 P05177 1/20 0.35
PKM P14618 1/20 0.35
TSHR P16473 1/20 0.35
NFKB1 P19838 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
GNAI1 P63096 1/20 0.35
PMP22 Q01453 1/20 0.35
KMT2A Q03164 1/20 0.35
HIF1A Q16665 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003372 0.92 PLA2G2A (0.38) OPRK1ACHECYP3A4CYP2C9MAPT
SCHEMBL2001936 0.90 OPRK1 (0.36) OPRK1FAAHCYP2C9ALDH1A1LMNA
SCHEMBL2004726 0.89 OPRK1 (0.42) OPRK1ACHECYP3A4CYP2C9ALDH1A1
SCHEMBL2002574 0.88 FAAH (0.42) OPRK1FAAHALDH1A1LMNAMAPT
SCHEMBL2003477 0.87 LMNA (0.40) OPRK1FAAHCYP3A4CYP2C9ALDH1A1
SCHEMBL2004659 0.87 KDM4E (0.37) OPRK1FAAHCYP3A4CYP2C9ALDH1A1
SCHEMBL2004340 0.86 F2RL3 (0.37) OPRK1FAAHLMNAMAPTALOX5AP
SCHEMBL2006197 0.86 ACHE (0.39) OPRK1ACHECYP3A4CYP2C9ALDH1A1
SCHEMBL2002529 0.85 PLA2G2A (0.43) CYP3A4CYP2C9ALDH1A1LMNAMAPT
SCHEMBL2004657 0.85 FAAH (0.38) OPRK1FAAHCYP3A4CYP2C9MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed