SCHEMBL4552391

SCHEMBL4552391

CS(=O)(=O)c1ccc(C(=O)C(N)CC(=O)O)cc1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.46
PTGS2 P35354 5/20 0.43
GSR P00390 2/20 0.43
GRM4 Q14833 1/20 0.43
GRIN2B Q13224 1/20 0.42
AKR1C2 P52895 1/20 0.41
AKR1C1 Q04828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2234923 0.77 CA2 (0.55)
SCHEMBL11133283 0.77 ALKBH5 (0.47)
SCHEMBL8506429 0.77 ALKBH5 (0.47)
SCHEMBL10708853 0.77 ALKBH5 (0.47)
Bromide SCHEMBL6489944 0.76 SLC7A5 (0.46)
SCHEMBL4552389 0.75 GSR (0.44) AKR1C3PTGS2GSRGRM4GRIN2B
SCHEMBL11235526 0.74 TAAR1 (0.49)
SCHEMBL5781468 0.74 EPHX2 (0.55) AKR1C3PTGS2AKR1C2AKR1C1
SCHEMBL20560043 0.73 ALDH1A1 (0.50)
SCHEMBL9539475 0.73 ALDH1A1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7638630-B2 Very Late Antigen-4 dependent inflammatory disease; asthma, allergic rhinitis, sinusitis, conjunctivitis, food allergy, inflammatory skin disorders, autoimmune disorders, or atherosclerosis, inflammatory skin disorder; methyl 3-[2-(2,6-dichlorophenyl)-6-quinolinyl]-2-hydroxy-2-propenoate UCB PHARMA S.A. (BE) 2009-12-29 US disclosed
US-20080064720-A1 2,6-Quinolinyl And 2,6-Naphthyl Derivatives, Processes For Preparing Them And Their Uses As Vla-4 Inhibitors UCB, S.A. (BE) 2008-03-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080064720-A1 2,6-Quinolinyl And 2,6-Naphthyl Derivatives, Processes For Preparing Them And Their Uses As Vla-4 Inhibitors VCAM1, HRH4, LTA4H AKR1C3 3272/4885PTGS2 1255/4885GSR 4751/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.