SCHEMBL4552389

SCHEMBL4552389

CS(=O)(=O)c1ccc(C(=O)C(CN)C(=O)O)cc1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSR P00390 2/20 0.44
AKR1C3 P42330 2/20 0.44
GRIN2B Q13224 1/20 0.43
PTGS2 P35354 3/20 0.43
ENPP2 Q13822 1/20 0.41
EPHX2 P34913 2/20 0.41
GRM4 Q14833 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8506427 0.76 MDM2 (0.59)
SCHEMBL4552391 0.75 AKR1C3 (0.46) GSRAKR1C3GRIN2BPTGS2GRM4
SCHEMBL8049079 0.74 ENPP2 (0.50) GSRAKR1C3PTGS2ENPP2
SCHEMBL15556865 0.73 GSR (0.59) GSRAKR1C3GRIN2BPTGS2ENPP2
SCHEMBL8722500 0.73 ENPP2 (0.48) GSRAKR1C3PTGS2ENPP2
SCHEMBL28427675 0.73 GSK3B (0.53) GSRAKR1C3PTGS2ENPP2
SCHEMBL8071790 0.72 GSR (0.46) GSRAKR1C3PTGS2ENPP2
SCHEMBL6510946 0.72 SRC (0.50) AKR1C3PTGS2
SCHEMBL34837 0.72 CA2 (0.61) GSRAKR1C3PTGS2ENPP2
Hydrochloric Acid SCHEMBL15465891 0.72 GSR (0.60) GSRAKR1C3GRIN2BPTGS2ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7638630-B2 Very Late Antigen-4 dependent inflammatory disease; asthma, allergic rhinitis, sinusitis, conjunctivitis, food allergy, inflammatory skin disorders, autoimmune disorders, or atherosclerosis, inflammatory skin disorder; methyl 3-[2-(2,6-dichlorophenyl)-6-quinolinyl]-2-hydroxy-2-propenoate UCB PHARMA S.A. (BE) 2009-12-29 US disclosed
US-20080064720-A1 2,6-Quinolinyl And 2,6-Naphthyl Derivatives, Processes For Preparing Them And Their Uses As Vla-4 Inhibitors UCB, S.A. (BE) 2008-03-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080064720-A1 2,6-Quinolinyl And 2,6-Naphthyl Derivatives, Processes For Preparing Them And Their Uses As Vla-4 Inhibitors VCAM1, HRH4, LTA4H GSR 4751/4885AKR1C3 3272/4885GRIN2B 2488/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.