SCHEMBL4573204

SCHEMBL4573204

NC(=O)C1(c2ccc(N3CCNCC3)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
USP2 O75604 1/20 0.49
TSHR P16473 1/20 0.49
HSD17B10 Q99714 1/20 0.49
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
ADRB1 P08588 6/20 0.46
HTR3E A5X5Y0 3/20 0.46
HTR3B O95264 3/20 0.46
HTR3A P46098 3/20 0.46
HTR3D Q70Z44 3/20 0.46
HTR3C Q8WXA8 3/20 0.46
SIGMAR1 Q99720 3/20 0.46
SIRT6 Q8N6T7 1/20 0.44
ACVR1 Q04771 1/20 0.43
ADRB2 P07550 1/20 0.42
NCF1 P14598 1/20 0.42
PLD1 Q13393 1/20 0.42
HTR6 P50406 1/20 0.42
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22471065 0.84 HSD11B1 (0.46) ALDH1A1USP2TSHRHSD17B10KDM4E
SCHEMBL18742793 0.79 HSD11B1 (0.48) ALDH1A1USP2TSHRHSD17B10KDM4E
SCHEMBL8110532 0.77 ADRB1 (0.54) ALDH1A1USP2TSHRHSD17B10KDM4E
SCHEMBL5572597 0.76 LMNA (0.55) ALDH1A1TSHRLMNASIGMAR1
SCHEMBL572738 0.75 ACVR1 (0.66) ALDH1A1USP2TSHRHSD17B10KDM4E
Hydrochloric Acid SCHEMBL3133889 0.73 ACVR1 (0.64) ALDH1A1USP2TSHRHSD17B10KDM4E
SCHEMBL4219088 0.73 OPRM1 (0.42) ALDH1A1KDM4ELMNA
SCHEMBL5570604 0.73 ADRB1 (0.77) ALDH1A1USP2TSHRHSD17B10KDM4E
Phenylpiperazine SCHEMBL2002893 0.73 ADRB1 (0.77) ALDH1A1USP2TSHRHSD17B10KDM4E
Tert-Butyl Formate SCHEMBL28033047 0.73 ADRB1 (0.39) ALDH1A1USP2TSHRHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed