SCHEMBL458252

SCHEMBL458252

CCc1ccc(-c2ccccc2Cl)cc1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
PAK1 Q13153 1/20 0.42
MAOB P27338 2/20 0.40
PGR P06401 1/20 0.40
GSK3B P49841 1/20 0.39
BACE1 P56817 1/20 0.39
TRPA1 O75762 1/20 0.39
CSNK2A2 P19784 1/20 0.39
CSNK2B P67870 1/20 0.39
CSNK2A1 P68400 1/20 0.39
CSNK2A3 Q8NEV1 1/20 0.39
ABL1 P00519 1/20 0.38
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
TYK2 P29597 1/20 0.38
JAK3 P52333 1/20 0.38
AOC3 Q16853 1/20 0.37
HSD11B1 P28845 1/20 0.37
AR P10275 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12653047 0.84 CYP2A6 (0.47) CYP2A6TNKS2PAK1MAOBPGR
SCHEMBL15060621 0.80 ALOX5AP (0.46) CYP2A6TNKS2PAK1MAOBPGR
SCHEMBL23956054 0.78 CSNK2A2 (0.43) CYP2A6TNKS2PAK1MAOBTRPA1
SCHEMBL455341 0.77 CRHBP (0.45)
SCHEMBL449516 0.75 ALOX5 (0.39) PGRGSK3BJAK2AOC3
SCHEMBL27875237 0.75 PDK1 (0.46) CYP2A6TNKS2PAK1
SCHEMBL9756794 0.73 CYP2A6 (0.42) CYP2A6TNKS2PGRBACE1TRPA1
SCHEMBL3031350 0.73 FASN (0.38)
SCHEMBL1623837 0.71 MAOB (0.61) CYP2A6MAOBCSNK2A2CSNK2BCSNK2A1
SCHEMBL9288019 0.70 TRPA1 (0.49) TRPA1CSNK2A2CSNK2BCSNK2A1CSNK2A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed