SCHEMBL458388

SCHEMBL458388

COc1cc(-c2ccccc2)ccc1I

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
TSHR P16473 2/20 0.45
HSD17B10 Q99714 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
CYP3A4 P08684 1/20 0.45
L3MBTL1 Q9Y468 3/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
KDM4E B2RXH2 5/20 0.44
HPGD P15428 5/20 0.44
MAPT P10636 3/20 0.44
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
USP2 O75604 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
ATM Q13315 1/20 0.44
LMNA P02545 1/20 0.43
GAA P10253 1/20 0.42
AAK1 Q2M2I8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4307124 0.89 ALDH1A1 (0.54) ALDH1A1TSHRHSD17B10TDP1CYP3A4
SCHEMBL4092939 0.84 KDM4E (0.47) ALDH1A1TSHRHSD17B10TDP1L3MBTL1
SCHEMBL4533772 0.81 L3MBTL1 (0.62) ALDH1A1TSHRHSD17B10TDP1L3MBTL1
SCHEMBL14305809 0.80 ALDH1A1 (0.45) ALDH1A1TSHRHSD17B10TDP1CYP3A4
SCHEMBL17400405 0.79 MAOA (0.47) ALDH1A1TSHRHSD17B10L3MBTL1NPC1
SCHEMBL4635995 0.78 KDM4E (0.50) ALDH1A1TSHRHSD17B10TDP1CYP3A4
SCHEMBL5961843 0.78 CYP3A4 (0.53) ALDH1A1TSHRHSD17B10TDP1CYP3A4
SCHEMBL358211 0.76 ALDH1A1 (0.80) ALDH1A1TSHRHSD17B10TDP1CYP3A4
SCHEMBL4839351 0.76 ACLY (0.52) ALDH1A1TSHRHSD17B10TDP1CYP3A4
SCHEMBL457121 0.76 DYRK1A (0.56) ALDH1A1TSHRHSD17B10TDP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed