SCHEMBL4586437

SCHEMBL4586437

CC(N)CCN1CCC(N(Cc2cccc(F)c2)c2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 8/20 0.47
OPRM1 P35372 7/20 0.45
TMEM97 Q5BJF2 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
CHRM2 P08172 1/20 0.38
CHRM3 P20309 1/20 0.38
UBE2M P61081 1/20 0.38
DCUN1D1 Q96GG9 1/20 0.38
KCNJ1 P48048 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586335 0.90 CCR5 (0.53) CCR5CHRM2CHRM3UBE2MDCUN1D1
SCHEMBL4586726 0.89 CCR5 (0.46) CCR5CHRM2CHRM3UBE2MDCUN1D1
SCHEMBL4586071 0.87 KCNH2 (0.52) CCR5DCUN1D1KCNJ1KCNH2
SCHEMBL4242144 0.84 UBE2M (0.43) CCR5UBE2MDCUN1D1
SCHEMBL4247149 0.80 UBE2M (0.42) CCR5OPRM1CHRM2CHRM3UBE2M
SCHEMBL4244706 0.76 GPR119 (0.50)
SCHEMBL4586432 0.75 CCR5 (0.54) CCR5
SCHEMBL4586423 0.75 CCR5 (0.41) CCR5OPRM1TMEM97
SCHEMBL4586731 0.73 OPRM1 (0.53) CCR5OPRM1CHRM2CHRM3
SCHEMBL4243399 0.73 CCR5 (0.53) CCR5UBE2MDCUN1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed