SCHEMBL4586726

SCHEMBL4586726

CC(N)CCN1CCC(N(Cc2cccc(Cl)c2)c2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 10/20 0.46
PGR P06401 1/20 0.44
CHRM2 P08172 1/20 0.40
CHRM3 P20309 1/20 0.40
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
ATM Q13315 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
UBE2M P61081 1/20 0.38
DCUN1D1 Q96GG9 1/20 0.38
HTR2A P28223 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
BACE1 P56817 1/20 0.38
DRD2 P14416 1/20 0.38
NPBWR1 P48145 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586335 0.90 CCR5 (0.53) CCR5CHRM2CHRM3UBE2MDCUN1D1
SCHEMBL4586437 0.89 CCR5 (0.47) CCR5CHRM2CHRM3UBE2MDCUN1D1
SCHEMBL4586071 0.87 KCNH2 (0.52) CCR5PGRDCUN1D1
SCHEMBL4243399 0.84 CCR5 (0.53) CCR5PGRUBE2MDCUN1D1
SCHEMBL4586764 0.82 CCR5 (0.51) CCR5PGRUBE2MDCUN1D1DRD2
SCHEMBL4586432 0.75 CCR5 (0.54) CCR5DRD2
SCHEMBL4241233 0.74 CCR5 (0.82) CCR5
SCHEMBL3814514 0.73 UBE2M (0.53) CCR5UBE2MDCUN1D1
SCHEMBL3820960 0.73 UBE2M (0.55) CCR5UBE2MDCUN1D1
SCHEMBL4586731 0.73 OPRM1 (0.53) CCR5CHRM2CHRM3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed