SCHEMBL4586335

SCHEMBL4586335

CC(N)CCN1CCC(N(Cc2ccccc2)c2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 12/20 0.53
DRD2 P14416 1/20 0.48
CHRM2 P08172 1/20 0.46
CHRM3 P20309 1/20 0.46
HTR2A P28223 2/20 0.45
UBE2M P61081 1/20 0.45
DCUN1D1 Q96GG9 1/20 0.45
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
BACE1 P56817 1/20 0.43
CCR2 P41597 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586437 0.90 CCR5 (0.47) CCR5CHRM2CHRM3UBE2MDCUN1D1
SCHEMBL4586726 0.90 CCR5 (0.46) CCR5DRD2CHRM2CHRM3HTR2A
SCHEMBL4586071 0.87 KCNH2 (0.52) CCR5DCUN1D1
SCHEMBL4586432 0.85 CCR5 (0.54) CCR5DRD2
SCHEMBL4586731 0.82 OPRM1 (0.53) CCR5DRD2CHRM2CHRM3
SCHEMBL4239263 0.82 CCR5 (0.49) CCR5CHRM2CHRM3UBE2MDCUN1D1
SCHEMBL4587113 0.80 CCR5 (0.57) CCR5DRD2UBE2MDCUN1D1
SCHEMBL4587621 0.78 CCR5 (0.55) CCR5DRD2UBE2MDCUN1D1
SCHEMBL4586715 0.78 CCR5 (0.55) CCR5DRD2UBE2MDCUN1D1
SCHEMBL4240396 0.74 ALDH1A1 (0.53) CCR5CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed