SCHEMBL4590241

SCHEMBL4590241

COc1ccc2ccc(=O)n3c2c1OCC3C=O

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
CYP19A1 P11511 1/20 0.32
NQO2 P16083 1/20 0.32
PTPRF P10586 1/20 0.32
LMNA P02545 2/20 0.32
MAPT P10636 1/20 0.32
KDM4E B2RXH2 3/20 0.31
HTR6 P50406 1/20 0.31
ALDH1A1 P00352 2/20 0.31
HSD17B10 Q99714 1/20 0.31
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30
HPGD P15428 1/20 0.30
ADRA1D P25100 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4590519 0.81 CNR1 (0.39) CNR1CNR2CYP19A1NQO2LMNA
SCHEMBL3227846 0.63 MTNR1A (0.31) CYP19A1NQO2MAPTALDH1A1
SCHEMBL4589655 0.63
SCHEMBL3110339 0.61 ALDH1A1 (0.40) CYP19A1NQO2MAPTKDM4EALDH1A1
SCHEMBL15875350 0.60 ADRA1A (0.35) CYP19A1NQO2MAPTKDM4EADRA1A
SCHEMBL5722849 0.58 LMNA (0.40) LMNAKDM4EALDH1A1HSD17B10HPGD
SCHEMBL2797396 0.58 HTR6 (0.47) CYP19A1NQO2MAPTKDM4EHTR6
SCHEMBL3106868 0.57 CYP19A1 (0.44) CYP19A1NQO2MAPTALDH1A1
SCHEMBL20549449 0.56 KCNH2 (0.35) KDM4EALDH1A1HSD17B10HPGD
SCHEMBL27877543 0.56 ACHE (0.57) CYP19A1LMNAMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008120003-A1 SUBSTITUTED PIPERIDINES FOR USE IN THE TREATMENT OF BACTERIAL INFECTIONS ASTRAZENECA AB (SE) 2008-10-09 WO disclosed