SCHEMBL4593251

SCHEMBL4593251

Cc1ccccc1C1(C(Cl)(Cl)C2(c3ccccc3C)N=NN=N2)N=NN=N1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
ACHE P22303 1/20 0.33
CYP3A4 P08684 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
HDAC4 P56524 1/20 0.31
PDK2 Q15119 1/20 0.31
CD44 P16070 1/20 0.30
OPRM1 P35372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593846 0.77 HTR2A (0.33) PDK2
SCHEMBL4593434 0.73 TSHR (0.35) TSHR
SCHEMBL19743353 0.72 PDK2 (0.43) TSHRACHECYP3A4TDP1PDK2
SCHEMBL8705403 0.69 TSHR (0.38) TSHRACHECYP3A4TDP1HDAC4
SCHEMBL4594159 0.69 ACHE (0.35) TSHRACHETDP1
SCHEMBL4593447 0.69 DRD1 (0.32)
SCHEMBL4593445 0.69 HDAC4 (0.34) TSHRACHECYP3A4TDP1HDAC4
SCHEMBL11470022 0.63 ACHE (0.45) TSHRACHECYP3A4TDP1HDAC4
O-Xylene SCHEMBL8518692 0.63 TSHR (0.71) TSHRACHECYP3A4TDP1
O-Xylene SCHEMBL6933035 0.62 TSHR (0.83) TSHRACHECYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937257-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES Nederlandse Organisatie voor toegepast- natuurwetenschappelijk onderzoek TNO (NL) 2008-07-02 EP disclosed
WO-2007037685-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2007-04-05 WO disclosed