SCHEMBL4596592

SCHEMBL4596592

O=C1NC[C@@](Cc2ccncc2)(c2ccccc2)N1C1CCNCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.36
SLC6A4 P31645 1/20 0.35
CYP3A4 P08684 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2D6 P10635 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP2C19 P33261 1/20 0.34
THPO P40225 1/20 0.34
TSHR P16473 2/20 0.34
KCNQ2 O43526 1/20 0.34
ALOX15 P16050 1/20 0.34
OPRM1 P35372 2/20 0.34
OPRL1 P41146 2/20 0.34
MAPK1 P28482 1/20 0.33
ATM Q13315 1/20 0.33
NSD3 Q9BZ95 1/20 0.33
CYP19A1 P11511 1/20 0.33
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4429230 0.78 MMP2 (0.35) CYP1A2TSHROPRM1OPRL1NSD3
SCHEMBL4597523 0.76 NPSR1 (0.32) ALDH1A1NSD3CHRM3GBA1
SCHEMBL5179386 0.74 GRIN1 (0.38) ALDH1A1ALOX15OPRM1NSD3CHRM2
SCHEMBL4598182 0.71 GRIN1 (0.36) SLC6A4CYP3A4CYP1A2ALDH1A1CYP2C19
Hydrochloric Acid SCHEMBL8413869 0.70 OPRM1 (0.35) CYP3A4ALDH1A1TSHROPRM1OPRL1
SCHEMBL4626507 0.69 NSD3 (0.36) ALDH1A1OPRM1ATMNSD3CHRM2
SCHEMBL4610698 0.69 NSD3 (0.36) ALDH1A1OPRM1ATMNSD3CHRM2
SCHEMBL4598539 0.69 NSD3 (0.34) SLC6A4CYP1A2ALDH1A1OPRM1OPRL1
SCHEMBL4415834 0.68 BACE1 (0.36) NSD3CHRM2CHRM3
SCHEMBL4595948 0.68 BACE1 (0.36) NSD3CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed