SCHEMBL4598182

SCHEMBL4598182

O=C1NC[C@](c2ccccc2)(c2ncccn2)N1C1CCNCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
NSD3 Q9BZ95 1/20 0.35
GRIN2B Q13224 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HTR1A P08908 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM3 P20309 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
PKM P14618 1/20 0.32
ALOX15 P16050 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
HRH1 P35367 1/20 0.32
KDM1A O60341 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5179386 0.89 GRIN1 (0.38) GRIN1GRIN2ANSD3GRIN2BKDM4E
SCHEMBL4598539 0.88 NSD3 (0.34) GRIN1GRIN2ANSD3GRIN2BKDM4E
SCHEMBL4597278 0.82 OPRL1 (0.33) GRIN1GRIN2ANSD3GRIN2BKDM4E
SCHEMBL4626507 0.73 NSD3 (0.36) NSD3KDM4ECHRM2CHRM3ALDH1A1
SCHEMBL4610698 0.73 NSD3 (0.36) NSD3KDM4ECHRM2CHRM3ALDH1A1
SCHEMBL4415834 0.72 BACE1 (0.36) GRIN1GRIN2ANSD3GRIN2BKDM4E
SCHEMBL4595948 0.72 BACE1 (0.36) GRIN1GRIN2ANSD3GRIN2BKDM4E
SCHEMBL2598433 0.71 HTR2C (0.40) GRIN1GRIN2ANSD3CHRM2CHRM3
SCHEMBL4597825 0.71 CHRM2 (0.39) GRIN2BHTR1ASLC6A4CHRM2CHRM3
SCHEMBL4596592 0.71 MMP13 (0.36) NSD3SLC6A4CHRM2CHRM3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed