SCHEMBL4598539

SCHEMBL4598539

O=C1NC[C@](c2ccccc2)(c2ccccn2)N1C1CCNCC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD3 Q9BZ95 1/20 0.34
GRIN1 Q05586 2/20 0.33
GRIN2A Q12879 2/20 0.33
CHRM2 P08172 2/20 0.33
CHRM3 P20309 2/20 0.33
GRIN2B Q13224 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
KDM4E B2RXH2 1/20 0.32
PLD1 Q13393 1/20 0.32
CXCR3 P49682 1/20 0.32
PLAT P00750 1/20 0.32
HTR1A P08908 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4598182 0.88 GRIN1 (0.36) NSD3GRIN1GRIN2ACHRM2CHRM3
SCHEMBL5179386 0.87 GRIN1 (0.38) NSD3GRIN1GRIN2ACHRM2CHRM3
SCHEMBL4597278 0.80 OPRL1 (0.33) NSD3GRIN1GRIN2AGRIN2BKDM4E
SCHEMBL4626507 0.71 NSD3 (0.36) NSD3CHRM2CHRM3KDM4EALDH1A1
SCHEMBL4610698 0.71 NSD3 (0.36) NSD3CHRM2CHRM3KDM4EALDH1A1
SCHEMBL4595948 0.70 BACE1 (0.36) NSD3GRIN1GRIN2ACHRM2CHRM3
SCHEMBL4415834 0.70 BACE1 (0.36) NSD3GRIN1GRIN2ACHRM2CHRM3
SCHEMBL4597825 0.69 CHRM2 (0.39) CHRM2CHRM3GRIN2BCHRM1HTR1A
SCHEMBL4596592 0.69 MMP13 (0.36) NSD3CHRM2CHRM3SLC6A4ALDH1A1
SCHEMBL4598352 0.68 SLC6A4 (0.41) PLATSLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed