SCHEMBL4597548

SCHEMBL4597548

O=C1NC2c3cccc(c3)C2(c2cccc(Cl)c2)N1C1CCNCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.36
TP53 P04637 3/20 0.35
MDM2 Q00987 3/20 0.35
DPP4 P27487 5/20 0.35
DPP9 Q86TI2 4/20 0.35
HTR6 P50406 3/20 0.35
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.35
HTR2B P41595 2/20 0.35
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35
CYP1A2 P05177 1/20 0.35
ADRB1 P08588 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR1A P08908 1/20 0.35
CYP2D6 P10635 1/20 0.35
THRB P10828 1/20 0.35
CYP2C9 P11712 1/20 0.35
SLC6A4 P31645 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4597529 0.69 BACE1 (0.38) DRD2TP53DPP4DPP9HTR6
SCHEMBL4596366 0.69 CHRM2 (0.37) DRD2TP53DPP4DPP9HTR6
SCHEMBL4596721 0.69 CHRM2 (0.37) DRD2TP53DPP4DPP9HTR6
SCHEMBL4597825 0.68 CHRM2 (0.39) DRD2TP53DPP4DPP9HTR6
SCHEMBL4596506 0.67 DRD2 (0.34) DRD2TP53DPP4DPP9HTR6
SCHEMBL4597256 0.67 DRD2 (0.34) DRD2TP53DPP4DPP9HTR6
SCHEMBL4598352 0.67 SLC6A4 (0.41) DRD2DPP4DPP9HTR6SLC6A4
SCHEMBL4597871 0.65 SLC6A2 (0.40) DRD2DPP4DPP9HTR6SLC6A4
SCHEMBL4597579 0.65 DRD2 (0.33) DRD2TP53DPP4DPP9HTR6
SCHEMBL4598045 0.64 SLC6A4 (0.43) DRD2DPP4DPP9HTR6SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed