SCHEMBL4598029

SCHEMBL4598029

O=C1NCCN1C1(c2cccc(F)c2)CCOCC1C1CCNCC1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 2/20 0.33
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
SLC6A9 P48067 4/20 0.32
OPRM1 P35372 4/20 0.32
OPRL1 P41146 2/20 0.31
HSD11B1 P28845 1/20 0.30
HTR6 P50406 1/20 0.30
USP2 O75604 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596509 0.88 CYP2C19 (0.34) PIK3C3ALDH1A1MEN1MAPTKMT2A
SCHEMBL4596047 0.88 SLC6A9 (0.36) ALDH1A1POLBSLC6A9OPRM1OPRL1
SCHEMBL4597794 0.79 HCRTR1 (0.31)
SCHEMBL4597761 0.69 KCNJ1 (0.44) ALDH1A1MAPTCYP2C19
SCHEMBL4597411 0.67
SCHEMBL4598373 0.66 GNAI3 (0.32)
SCHEMBL4598027 0.65 CHRNA1 (0.32) ALDH1A1KDM4EMEN1POLBMAPT
SCHEMBL3900550 0.62 USP2 (0.38) ALDH1A1SLC6A9OPRM1OPRL1HSD11B1
SCHEMBL3910153 0.59 OPRM1 (0.40) ALDH1A1MEN1KMT2ASLC6A9OPRM1
SCHEMBL3860581 0.58 ALDH1A1 (0.43) ALDH1A1POLBSLC6A9OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed