SCHEMBL4601338

SCHEMBL4601338

C=CC(=O)Oc1c(OCCOC)cccc1OS(=O)(=O)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.42
RXFP1 Q9HBX9 3/20 0.37
HTT P42858 2/20 0.36
THRB P10828 2/20 0.35
DRD2 P14416 3/20 0.34
DRD1 P21728 2/20 0.34
DRD4 P21917 2/20 0.34
DRD5 P21918 2/20 0.34
DRD3 P35462 2/20 0.34
KDM4E B2RXH2 2/20 0.34
THRA P10827 1/20 0.33
KMT2A Q03164 1/20 0.33
ITK Q08881 1/20 0.33
HTR2A P28223 1/20 0.32
GRM2 Q14416 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4601601 0.81 EGFR (0.47) EGFRRXFP1HTTTHRBKDM4E
SCHEMBL4602183 0.79 EGFR (0.47) EGFRTHRBKMT2A
SCHEMBL4600130 0.77 EGFR (0.47) EGFRRXFP1HTTTHRBKDM4E
SCHEMBL4601033 0.76 EGFR (0.44) EGFRTHRBKDM4ETHRAHTR2A
SCHEMBL4602169 0.76 EGFR (0.41) EGFRRXFP1HTTKDM4EKMT2A
SCHEMBL27360839 0.75 THRB (0.42) THRBDRD2DRD1DRD4DRD5
SCHEMBL4601218 0.74 MRGPRX4 (0.46) EGFRRXFP1HTTKDM4EKMT2A
SCHEMBL4600628 0.74 EGFR (0.47) EGFRTHRBKDM4ETHRAKMT2A
SCHEMBL4601685 0.74 RXFP1 (0.48) EGFRRXFP1HTTKDM4EKMT2A
SCHEMBL4600843 0.74 RAB9A (0.50) EGFRHTTKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912645-A2 THERAPEUTIC AGENT FOR DIABETES Takeda Pharmaceutical Company Limited (JP) 2008-04-23 EP disclosed
WO-2007018314-A2 THERAPEUTIC AGENT FOR DIABETES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-15 WO disclosed