SCHEMBL4621655

SCHEMBL4621655

[c]1cccc(-c2ccccc2)c1-c1ccc(-c2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
HSD17B10 Q99714 3/20 0.38
BCL2L1 Q07817 2/20 0.38
MAPK1 P28482 2/20 0.38
HPGD P15428 1/20 0.38
CYP2A6 P11509 1/20 0.38
TDP1 Q9NUW8 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
MMP3 P08254 1/20 0.36
ALOX5 P09917 1/20 0.35
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
PTGS2 P35354 1/20 0.35
MEN1 O00255 1/20 0.35
APAF1 O14727 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL185890 0.96 ALDH1A1 (0.41) ALDH1A1HSD17B10BCL2L1MAPK1HPGD
SCHEMBL9559797 0.91 PTGS2 (0.39) BCL2L1PTGS2MEN1MAPTKMT2A
SCHEMBL28716480 0.88 CYP1A2 (0.50) ALDH1A1CYP2A6CYP1A2PTGS2MEN1
SCHEMBL9559722 0.88 PTGS2 (0.40) ALDH1A1HSD17B10BCL2L1HPGDPTGS2
SCHEMBL7754417 0.87 ALDH1A1 (0.38) ALDH1A1HSD17B10BCL2L1MAPK1HPGD
SCHEMBL3327939 0.86 MAOA (0.38) ALDH1A1HSD17B10BCL2L1MAPK1HPGD
SCHEMBL7703864 0.85 GSTP1 (0.49) PTGS2NPC1RAB9A
SCHEMBL28598863 0.84 NOTUM (0.50) ALDH1A1MAPK1NPC1MAPTHTT
SCHEMBL28592124 0.84 NOTUM (0.50) ALDH1A1MAPK1NPC1MAPTHTT
SCHEMBL11032010 0.84 MAPT (0.40) HPGDCYP2A6CYP1A2PTGS2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1897880-A1 1,3-BENZOTHIAZINONE DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2008-03-12 EP disclosed