SCHEMBL4630907

SCHEMBL4630907

C[C@H](NC(=O)OC(C)(C)CCc1ccccc1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.52
TSHR P16473 1/20 0.52
KMT2A Q03164 1/20 0.52
NAAA Q02083 1/20 0.48
ACE P12821 2/20 0.45
ATM Q13315 1/20 0.45
CTSK P43235 4/20 0.44
CTSS P25774 1/20 0.44
LTA4H P09960 2/20 0.44
MME P08473 1/20 0.44
PPARA Q07869 2/20 0.43
PPARG P37231 1/20 0.43
PRSS1 P07477 1/20 0.42
CTSG P08311 1/20 0.42
CTRB1 P17538 1/20 0.42
CMA1 P23946 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18342073 0.83 NAAA (0.46) MEN1KMT2ANAAAATMCTSK
SCHEMBL5340682 0.81 PPARA (0.52) MEN1TSHRKMT2AATMCTSK
SCHEMBL18342075 0.79 NAAA (0.45) MEN1TSHRKMT2ANAAAATM
SCHEMBL5144290 0.78 NAAA (0.43) MEN1TSHRKMT2ANAAAPPARA
SCHEMBL3504292 0.78 NAAA (0.44) TSHRKMT2ANAAASMN1; SMN2
SCHEMBL5145960 0.77 NPC1 (0.45) NAAAATM
SCHEMBL3834968 0.77 SIGMAR1 (0.46) NAAAACECTSKCTSS
SCHEMBL8982552 0.76 NAAA (0.44) NAAACTSKCTSS
SCHEMBL873380 0.76 ALDH1A1 (0.48) MEN1KMT2ANAAASMN1; SMN2
SCHEMBL25054029 0.76 CTSS (0.69) ACECTSKCTSSPPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1922306-A2 AMIDE DERIVATIVES AS ROCK INHIBITORS Astellas Pharma Inc. (JP) 2008-05-21 EP disclosed
WO-2007026920-A2 AMIDE DERIVATIVES AS ROCK INHIBITORS ASTELLAS PHARMA INC. (JP) 2007-03-08 WO disclosed