SCHEMBL4632782

SCHEMBL4632782

CC(C)(C)OC(=O)N(CCO)c1cccc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
LTB4R2 Q9NPC1 2/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
HDAC6 Q9UBN7 3/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC5 Q9UQL6 1/20 0.41
MAPT P10636 2/20 0.41
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
F2 P00734 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
RXFP1 Q9HBX9 2/20 0.39
CETP P11597 1/20 0.39
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1969523 0.87 CACNA1G (0.40) F2CETP
SCHEMBL4499074 0.85 LTB4R2 (0.45) MEN1KMT2ALTB4R2CYP1A2CYP3A4
SCHEMBL10670515 0.82 LTB4R2 (0.44) MEN1KMT2ALTB4R2CYP1A2CYP3A4
SCHEMBL9525464 0.82 ALDH1A1 (0.43) KMT2ALTB4R2MAPTGAAHTT
SCHEMBL30797543 0.82 ALDH1A1 (0.43) KMT2ALTB4R2MAPTGAAHTT
SCHEMBL10401421 0.82 MTNR1A (0.40) KMT2AHDAC6HDAC1MAPTF2
SCHEMBL9738368 0.81 LTB4R2 (0.44) MEN1KMT2ALTB4R2CYP1A2CYP3A4
SCHEMBL4437768 0.81 MEN1 (0.54) MEN1KMT2ALTB4R2CYP1A2CYP3A4
SCHEMBL1624311 0.81 SMN1; SMN2 (0.51) MEN1KMT2ACYP3A4CYP2C19HDAC6
SCHEMBL440958 0.80 RXFP1 (0.43) LTB4R2CYP1A2CYP3A4CYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888538-A1 (3,4-DIHYDRO-QUINAZOLIN-2-YL)-(2-ARYLOXY-ETHYL)-AMINES HAVING AN ACTIVITY ON THE 5-HT RECEPTOR F. Hoffmann-Roche AG (CH) 2008-02-20 EP disclosed
WO-2006117305-A1 (3,4-DIHYDRO-QUINAZOLIN-2-YL)-(2-ARYLOXY-ETHYL)-AMINES HAVING AN ACTIVITY ON THE 5-HT RECEPTOR F. HOFFMANN-LA ROCHE AG (CH) 2006-11-09 WO disclosed