SCHEMBL4634337

SCHEMBL4634337

CN(C)CC1(Cc2ccc(F)cc2)CCN(C(=O)O)CC1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.43
OPRL1 P41146 3/20 0.43
HSD11B1 P28845 1/20 0.40
KMT2A Q03164 1/20 0.38
AGTR2 P50052 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
KDM1A O60341 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5674689 0.83 MEN1 (0.45) KMT2AKDM1A
SCHEMBL4634957 0.78 HSD11B1 (0.44) OPRL1HSD11B1KMT2AKDM1A
SCHEMBL4634537 0.77 CYP46A1 (0.50) OPRM1OPRL1HSD11B1OPRD1OPRK1
SCHEMBL4634991 0.76 HSD11B1 (0.41) HSD11B1KMT2A
Hydrochloric Acid SCHEMBL5810883 0.75 HSD11B1 (0.43) HSD11B1KDM1A
SCHEMBL4635399 0.75 KDM1A (0.41) OPRM1OPRL1HSD11B1KMT2AOPRK1
SCHEMBL4633737 0.74 OPRD1 (0.39) OPRM1KMT2AOPRD1KDM1A
SCHEMBL5807513 0.74 HTT (0.41) HSD11B1
SCHEMBL4634641 0.73 ALDH1A1 (0.41)
SCHEMBL2798597 0.73 ALDH1A1 (0.43) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928829-A1 PIPERIDINE DERIVATIVES AS ANTAGONISTS OF THE CC CHEMOKINE RECEPTOR CCR1 AND THEIR USE AS ANTI-INFLAMMATORY AGENTS Schering Aktiengesellschaft (DE) 2008-06-11 EP disclosed
WO-2006066948-A1 PIPERIDINE DERIVATIVES AS ANTAGONISTS OF THE CC CHEMOKINE RECEPTOR CCR1 AND THEIR USE AS ANTI-INFLAMMATORY AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 2006-06-29 WO disclosed