SCHEMBL4649332

SCHEMBL4649332

Cc1cccc([N+](C)(C)Cc2ccccc2)c1Br

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
MAPT P10636 1/20 0.35
DNM1 Q05193 2/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TP53 P04637 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 2/20 0.33
TSHR P16473 2/20 0.31
SCN4A P35499 1/20 0.31
MCHR1 Q99705 1/20 0.31
SCN8A Q9UQD0 1/20 0.30
HTR7 P34969 1/20 0.30
LMNA P02545 1/20 0.30
CYP2D6 P10635 1/20 0.30
TAS2R10 Q9NYW0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL5117868 0.98 ALDH1A1 (0.41) ALDH1A1KDM4ETDP1MAPTDNM1
SCHEMBL564456 0.83 ALDH1A1 (0.50) ALDH1A1KDM4ETDP1DNM1MEN1
Hydrochloric Acid SCHEMBL31362231 0.82 ALDH1A1 (0.54) ALDH1A1KDM4ETDP1DNM1MEN1
SCHEMBL4649848 0.78 ALDH1A1 (0.48) ALDH1A1KDM4ETDP1DNM1MEN1
Bromide SCHEMBL5127809 0.77 ALDH1A1 (0.47) ALDH1A1KDM4ETDP1DNM1MEN1
SCHEMBL28423034 0.73 KDM4E (0.47) ALDH1A1KDM4ETDP1DNM1MEN1
Trifluoromethanesulfonic Acid SCHEMBL565377 0.72 GPR3 (0.36) ALDH1A1KDM4ETDP1
SCHEMBL28256353 0.71 ALDH1A1 (0.48) ALDH1A1KDM4ETDP1DNM1MEN1
SCHEMBL4649328 0.70 GABRA1 (0.36) ALDH1A1KDM4ETDP1MAPTMAPK1
Bromide SCHEMBL11060577 0.69 ALDH1A1 (0.47) ALDH1A1KDM4ETDP1DNM1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966138-A2 SUBSTITUTED TRICYCLIC PIPERIDONE DERIVATIVES Grünenthal GmbH (DE) 2008-09-10 EP disclosed
WO-2007079929-A2 SUBSTITUTED TRICYCLIC PIPERIDONE DERIVATIVES Grünenthal GmbH (DE) 2007-07-19 WO disclosed