SCHEMBL4650586

SCHEMBL4650586

O=S(=O)(c1ccccc1)c1cnc2ccc(OCCN3CCCCC3)cc2c1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 5/20 0.50
HRH3 Q9Y5N1 9/20 0.49
BACE1 P56817 1/20 0.49
KCNH2 Q12809 1/20 0.49
ADORA2A P29274 1/20 0.48
ADORA1 P30542 1/20 0.48
TLR9 Q9NR96 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4650105 1.00 LTA4H (0.50) LTA4HHRH3BACE1KCNH2ADORA2A
SCHEMBL4649999 0.95 TLR9 (0.54) HRH3KCNH2TLR9
SCHEMBL4649201 0.91 ADORA3 (0.50) LTA4HADORA2AADORA1
SCHEMBL4649413 0.79 KDM4E (0.52) LTA4HADORA2AADORA1
SCHEMBL4649409 0.79 CHRNB2 (0.56)
SCHEMBL4650585 0.78 HTR6 (0.52) HRH3BACE1
SCHEMBL4649915 0.78 HTR6 (0.52) HRH3BACE1
SCHEMBL4649244 0.77 HTR6 (0.53) LTA4HHRH3
SCHEMBL3535866 0.77 HRH3 (0.51) LTA4HHRH3BACE1KCNH2ADORA2A
SCHEMBL2814385 0.77 LTA4H (0.55) LTA4HHRH3TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730112-B1 3-((HETERO)ARYLSULFONYL)-8'[ (AMINOALKYL)OXY]QUINOLINES AS 5-HT6 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF CNS DISORDERS GLAXO GROUP LTD (GB) 2008-09-03 EP claimed