SCHEMBL4658162

SCHEMBL4658162

CON1c2ccc(OC(F)(F)F)cc2C(C)(C)[C@H]2COc3ccccc3[C@H]21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 2/20 0.36
HSPA9 P38646 2/20 0.33
GAA P10253 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CTSD P07339 1/20 0.33
BACE1 P56817 1/20 0.33
SLC6A4 P31645 1/20 0.32
TMEM97 Q5BJF2 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
HCRTR1 O43613 1/20 0.32
KCNH2 Q12809 2/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
P2RY1 P47900 1/20 0.32
ABCB1 P08183 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TACR1 P25103 1/20 0.31
CHRM5 P08912 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4564019 0.85 LMNA (0.38) HCRTR2GAAL3MBTL1ALDH1A1CTSD
SCHEMBL4564341 0.84 HSD11B1 (0.39) LMNA
SCHEMBL4564085 0.84 HSP90AA1 (0.39) GAAL3MBTL1ALDH1A1HSP90AA1
SCHEMBL4657250 0.82 LMNA (0.38) HCRTR2GAAL3MBTL1ALDH1A1CTSD
SCHEMBL4657674 0.82 NR1H3 (0.37) GAAL3MBTL1ALDH1A1LMNA
SCHEMBL4629499 0.82 HSP90AA1 (0.39) GAAL3MBTL1ALDH1A1LMNAHSP90AA1
SCHEMBL4556263 0.81 ALDH1A1 (0.37) GAAL3MBTL1ALDH1A1NPSR1LMNA
SCHEMBL4627927 0.81 ALDH1A1 (0.37) GAAL3MBTL1ALDH1A1NPSR1LMNA
SCHEMBL4564158 0.81 HTR2B (0.36) GAAL3MBTL1ALDH1A1BACE1TMEM97
SCHEMBL4564188 0.80 LTB4R (0.34) GAAL3MBTL1ALDH1A1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907395-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2008-04-09 EP claimed
WO-2007002867-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2007-01-04 WO claimed
EP-1907395-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2008-04-09 EP disclosed
WO-2007002867-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2007-01-04 WO disclosed