SCHEMBL4659306

SCHEMBL4659306

O=C(CNC(=O)O)Cc1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.50
MEN1 O00255 4/20 0.50
ALDH1A1 P00352 3/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
CTBP2 P56545 1/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
HPGD P15428 1/20 0.47
L3MBTL1 Q9Y468 4/20 0.46
LMNA P02545 1/20 0.46
CNR2 P34972 2/20 0.45
CNR1 P21554 1/20 0.45
MAPT P10636 1/20 0.44
EGFR P00533 2/20 0.44
ERBB2 P04626 2/20 0.44
ERCC1 P07992 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4659431 0.83 L3MBTL1 (0.54) KMT2AMEN1ALDH1A1NPC1RAB9A
SCHEMBL4582402 0.82 CES1 (0.52) KMT2AMEN1ALDH1A1RAB9ACYP2C9
SCHEMBL7965958 0.81 RAB9A (0.51) KMT2AALDH1A1NPC1RAB9ACTBP2
SCHEMBL4662034 0.81 TACR1 (0.40) KMT2AMEN1ALDH1A1RAB9ACTBP2
SCHEMBL1479915 0.80 NPC1 (0.55) KMT2AMEN1ALDH1A1NPC1RAB9A
SCHEMBL4327956 0.79 CTBP2 (0.52) KMT2AMEN1ALDH1A1NPC1RAB9A
SCHEMBL4660490 0.77 HTT (0.57) KMT2AALDH1A1NPC1RAB9ACTBP2
SCHEMBL28297938 0.77 KMT2A (0.49) KMT2AMEN1ALDH1A1RAB9ACYP2C9
SCHEMBL4768501 0.77 NR1H4 (0.54) ALDH1A1RAB9ALMNAMAPT
SCHEMBL8406795 0.76 L3MBTL1 (0.66) KMT2AMEN1ALDH1A1CTBP2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2004166-A2 INHIBITORS OF SEMICARBAZIDE-SENSITIVE AMINE OXIDASE (SSAO) AND VAP-1 MEDIATED ADHESION USEFUL FOR TREATMENT AND PREVENTION OF DISEASES LA JOLLA PHARMACEUTICAL COMPANY (US) 2008-12-24 EP disclosed
WO-2007120528-A2 INHIBITORS OF SEMICARBAZIDE-SENSITIVE AMINE OXIDASE (SSAO) AND VAP-1 MEDIATED ADHESION USEFUL FOR TREATMENT AND PREVENTION OF DISEASES LA JOLLA PHARMACEUTICAL COMPANY (US) 2007-10-25 WO disclosed