SCHEMBL4582402

SCHEMBL4582402

O=C(CNC(=O)O)Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.52
CES2 O00748 1/20 0.52
AKR1B1 P15121 1/20 0.52
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
TSHR P16473 1/20 0.48
CYP2C19 P33261 1/20 0.48
EPHX2 P34913 1/20 0.47
HPGD P15428 3/20 0.46
ALDH1A1 P00352 3/20 0.46
GAA P10253 2/20 0.46
ATM Q13315 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7527957 0.84 CES2 (0.48) CES1CES2AKR1B1MEN1KMT2A
SCHEMBL4659431 0.84 L3MBTL1 (0.54) MEN1KMT2ATDP1L3MBTL1HPGD
SCHEMBL7965958 0.82 RAB9A (0.51) KMT2ATDP1CYP2D6CYP2C9CYP2C19
SCHEMBL4659306 0.82 KMT2A (0.50) MEN1KMT2ATDP1L3MBTL1CYP1A2
SCHEMBL4659414 0.82 CTBP2 (0.54) MEN1KMT2AL3MBTL1HPGDALDH1A1
SCHEMBL24487008 0.81 CES2 (0.45) CES1CES2AKR1B1MEN1KMT2A
SCHEMBL5150815 0.81 HDAC8 (0.57) CES1CES2AKR1B1MEN1KMT2A
SCHEMBL4660680 0.81 RAB9A (0.49) ALDH1A1RAB9A
SCHEMBL10962854 0.80 VNN1 (0.56) CES1CES2AKR1B1MEN1KMT2A
SCHEMBL51367 0.80 CES1 (0.64) CES1CES2AKR1B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968568-A2 INHIBITORS OF Akt ACTIVITY SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007076423-A2 INHIBITORS OF Akt ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed