SCHEMBL4674253

SCHEMBL4674253

c1cncc(COc2ccc(N3CCNCC3)cc2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.59
NMT1 P30419 1/20 0.53
CHRNB2 P17787 2/20 0.51
CHRNA4 P43681 2/20 0.51
ALDH1A1 P00352 2/20 0.51
PRMT5 O14744 1/20 0.49
LTA4H P09960 1/20 0.48
PDE3B Q13370 1/20 0.48
PDE3A Q14432 1/20 0.48
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
ADRB1 P08588 1/20 0.47
HTR3A P46098 1/20 0.47
HTR3D Q70Z44 1/20 0.47
HTR3C Q8WXA8 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
ADRB2 P07550 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4674249 0.85 MAPK1 (0.47) HTR6LTA4HFGFR1MAPK1PRKDC
SCHEMBL4676367 0.83 ADRB2 (0.60) PRMT5LTA4HHTR3EHTR3BADRB1
SCHEMBL335477 0.83 LTA4H (0.64) HTR6ALDH1A1PRMT5LTA4HMAPT
Hydrochloric Acid SCHEMBL2156238 0.82 LTA4H (0.62) HTR6ALDH1A1PRMT5LTA4HMAPT
SCHEMBL28048524 0.80 MAPK1 (0.64) ALDH1A1HTTMAPK1CYP19A1CYP11B1
SCHEMBL5230479 0.78 LTA4H (0.57) HTR6CHRNB2CHRNA4ALDH1A1PRMT5
SCHEMBL6014772 0.78 HTR6 (0.58) HTR6NMT1CHRNB2CHRNA4PDE3B
SCHEMBL905960 0.76 HTR2C (0.70) HTR6NMT1CHRNB2CHRNA4ALDH1A1
SCHEMBL29664303 0.76 HTR6 (0.58) HTR6NMT1CHRNB2CHRNA4ALDH1A1
SCHEMBL6100222 0.76 HTR6 (0.58) HTR6NMT1CHRNB2CHRNA4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0958287-B2 SULFAMIDE-METALLOPROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2008-04-09 EP disclosed
EP-0958287-B1 SULFAMIDE-METALLOPROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2002-09-11 EP disclosed