SCHEMBL4690210

SCHEMBL4690210

NC(=O)c1ccccc1[CH]CCN1CC2CN(C(=O)c3c(N)cccc3C(F)(F)F)C[C@@H]2C1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RBP4 P02753 5/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP3A4 P08684 1/20 0.35
SLC6A1 P30531 4/20 0.35
CCR5 P51681 7/20 0.34
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
PARP1 P09874 1/20 0.33
CCL5 P13501 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691301 0.84 HCRTR1 (0.44) CYP2C9CYP2C19CCR5HCRTR1HCRTR2
SCHEMBL4691802 0.82 CCR5 (0.48) SLC6A1CCR5HCRTR1HCRTR2
SCHEMBL4691673 0.81 HCRTR1 (0.38) CCR5HCRTR1HCRTR2CCL5
SCHEMBL3284141 0.80 CCR5 (0.42) SLC6A1CCR5HCRTR1HCRTR2
SCHEMBL4694455 0.79 CHRNB2 (0.44) RBP4CCR5
SCHEMBL4689903 0.78 P2RX7 (0.41) CYP2C9CYP2C19SLC6A1CCR5
SCHEMBL4691928 0.77 MAPK1 (0.41) HCRTR1HCRTR2
SCHEMBL4695175 0.76 CCR5 (0.47) RBP4CCR5CCL5
SCHEMBL4694309 0.76 HCRTR1 (0.39) HCRTR1HCRTR2
SCHEMBL4693059 0.75 CCR5 (0.37) SLC6A1CCR5PARP1CCL5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed