SCHEMBL4689903

SCHEMBL4689903

NC(=O)c1ccccc1[CH]CCN1CC2CN(C(=O)c3ccccc3Cl)C[C@@H]2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.41
RAB9A P51151 2/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
CCR5 P51681 2/20 0.39
KCNA5 P22460 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTR2B P41595 1/20 0.39
MAPK14 Q16539 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
THRB P10828 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691802 0.92 CCR5 (0.48) RAB9AKMT2AMEN1CCR5SLC6A1
SCHEMBL4694336 0.89 HCRTR1 (0.36) CCR5THRBALDH1A1
SCHEMBL3284141 0.87 CCR5 (0.42) KMT2AMEN1CCR5SLC6A1
SCHEMBL4694455 0.87 CHRNB2 (0.44) KMT2AMEN1CCR5ALDH1A1HPGD
SCHEMBL4694264 0.86 ALDH1A1 (0.36) CCR5SLC6A1ALDH1A1
SCHEMBL4693059 0.84 CCR5 (0.37) KMT2AMEN1CCR5SLC6A1ALDH1A1
SCHEMBL4691301 0.83 HCRTR1 (0.44) CCR5CYP2C9CYP2C19LMNAHTT
SCHEMBL4692078 0.83 CCR5 (0.40) CCR5SLC6A1
SCHEMBL4693208 0.83 CCR5 (0.42) CCR5
SCHEMBL4694309 0.83 HCRTR1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed