SCHEMBL4694455

SCHEMBL4694455

NC(=O)c1ccccc1[CH]CCN1CC2CN(C(=O)c3ccccc3)C[C@@H]2C1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.44
CHRNB4 P30926 3/20 0.44
CHRNA3 P32297 3/20 0.44
CHRNA7 P36544 3/20 0.44
CHRNA4 P43681 3/20 0.44
CCR5 P51681 4/20 0.39
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KCNH2 Q12809 1/20 0.36
PLA2G1B P04054 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
PTPN1 P18031 1/20 0.35
RBP4 P02753 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691928 0.89 MAPK1 (0.41) SMN1; SMN2ALDH1A1HPGD
SCHEMBL4690512 0.89 ALDH1A1 (0.43) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL4690222 0.87 CHRNA4 (0.46) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL4689903 0.87 P2RX7 (0.41) CCR5MEN1KMT2AALDH1A1HPGD
SCHEMBL4696365 0.86 GRM5 (0.38) CCR5ALDH1A1
SCHEMBL4691301 0.85 HCRTR1 (0.44) CCR5
SCHEMBL4691802 0.85 CCR5 (0.48) CCR5MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL4693059 0.84 CCR5 (0.37) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL4693659 0.84 CHRNB2 (0.47) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL3282844 0.84 GRIN2B (0.44) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed