SCHEMBL4690512

SCHEMBL4690512

N#Cc1ccc(C(=O)N2CC3CN(CC[CH]c4ccccc4C(N)=O)C[C@H]3C2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
KCNA5 P22460 1/20 0.39
FASN P49327 1/20 0.38
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
KDM1A O60341 3/20 0.35
MGLL Q99685 1/20 0.35
SLC6A7 Q99884 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
PRKAB2 O43741 1/20 0.34
PRKAG1 P54619 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAA1 Q13131 1/20 0.34
PRKAG3 Q9UGI9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4696365 0.90 GRM5 (0.38) ALDH1A1KCNA5HCRTR1HCRTR2GRIN2B
SCHEMBL4694455 0.89 CHRNB2 (0.44) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4690222 0.81 CHRNA4 (0.46) ALDH1A1HCRTR1HCRTR2MAPTCHRNB2
SCHEMBL4689903 0.81 P2RX7 (0.41) ALDH1A1KCNA5
SCHEMBL4691928 0.80 MAPK1 (0.41) ALDH1A1HCRTR1HCRTR2GRIN2B
SCHEMBL4691802 0.79 CCR5 (0.48) ALDH1A1HCRTR1HCRTR2
SCHEMBL4691301 0.79 HCRTR1 (0.44) HCRTR1HCRTR2
SCHEMBL4693059 0.78 CCR5 (0.37) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4693659 0.78 CHRNB2 (0.47) ALDH1A1MAPTCHRNB2CHRNB4CHRNA3
SCHEMBL4695117 0.78 HDAC3 (0.41) HCRTR1HCRTR2CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed