SCHEMBL4690222

SCHEMBL4690222

NC(=O)c1ccccc1[CH]CCN1CC2CN(C(=O)c3ccoc3)C[C@@H]2C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA4 P43681 3/20 0.46
CHRNB2 P17787 2/20 0.46
CHRNB4 P30926 2/20 0.46
CHRNA3 P32297 2/20 0.46
CHRNA7 P36544 2/20 0.46
CCR5 P51681 3/20 0.43
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
PARP1 P09874 1/20 0.32
MAPT P10636 1/20 0.32
RECQL P46063 1/20 0.32
GPR52 Q9Y2T5 1/20 0.32
POLB P06746 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
NAMPT P43490 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694455 0.87 CHRNB2 (0.44) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4693659 0.83 CHRNB2 (0.47) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4689903 0.81 P2RX7 (0.41) CCR5ALDH1A1MEN1KMT2APOLB
SCHEMBL4691928 0.81 MAPK1 (0.41) ALDH1A1HCRTR1HCRTR2
SCHEMBL4690512 0.81 ALDH1A1 (0.43) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4695594 0.80 HCRTR1 (0.36) CHRNA4CCR5HCRTR1HCRTR2
SCHEMBL4691802 0.80 CCR5 (0.48) CCR5ALDH1A1MEN1KMT2AHCRTR1
SCHEMBL4691301 0.80 HCRTR1 (0.44) CCR5HCRTR1HCRTR2
SCHEMBL4696365 0.79 GRM5 (0.38) CCR5ALDH1A1HCRTR1HCRTR2PARP1
SCHEMBL4693059 0.79 CCR5 (0.37) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed