SCHEMBL4691604

SCHEMBL4691604

Cc1nc(C(=O)N2CC3CN(C(CC(N)=O)c4ccc(C)c(Cl)c4)CC3C2)cs1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GFER P55789 1/20 0.42
CHRM2 P08172 3/20 0.37
CHRM3 P20309 3/20 0.37
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
KCNH2 Q12809 2/20 0.35
TNF P01375 1/20 0.34
GRM5 P41594 1/20 0.34
ALK Q9UM73 1/20 0.34
TRPC3 Q13507 3/20 0.33
TRPC6 Q9Y210 3/20 0.33
KMT2A Q03164 2/20 0.33
HRH4 Q9H3N8 1/20 0.33
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691532 0.85 CHRNB2 (0.44) HCRTR1HCRTR2TNF
SCHEMBL4695666 0.83 SMN1; SMN2 (0.42) GFERHCRTR1HCRTR2TNFHRH4
SCHEMBL4694340 0.83 TNF (0.36) CHRM2HCRTR1HCRTR2TNFKMT2A
SCHEMBL4693800 0.82 RAB9A (0.43) HCRTR1HCRTR2TNFKMT2AMEN1
SCHEMBL4695972 0.82 CHRNB2 (0.40) GFERHCRTR1HCRTR2TNFKMT2A
SCHEMBL4694328 0.82 TNF (0.35) CHRM2CHRM3HCRTR1HCRTR2TNF
SCHEMBL4694334 0.81 HCRTR1 (0.43) HCRTR1HCRTR2TNF
SCHEMBL3281863 0.81 HCRTR1 (0.48) HCRTR1HCRTR2KCNH2TNF
SCHEMBL4690403 0.81 HCRTR1 (0.39) HCRTR1HCRTR2TNFHRH4
SCHEMBL4694248 0.81 ALDH1A1 (0.39) HCRTR1HCRTR2TNFKMT2AHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed