SCHEMBL4694340

SCHEMBL4694340

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4sccc4Cl)CC3C2)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HCRTR1 O43613 4/20 0.35
HCRTR2 O43614 4/20 0.35
CHRM2 P08172 1/20 0.34
HTR1A P08908 1/20 0.34
S1PR1 P21453 1/20 0.33
RAB9A P51151 1/20 0.32
HRH2 P25021 1/20 0.32
HRH1 P35367 1/20 0.32
LMNA P02545 1/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
SLC6A3 Q01959 2/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694328 0.84 TNF (0.35) TNFALDH1A1HCRTR1HCRTR2CHRM2
SCHEMBL4694334 0.83 HCRTR1 (0.43) TNFHCRTR1HCRTR2CCR5
SCHEMBL4690403 0.83 HCRTR1 (0.39) TNFALDH1A1HCRTR1HCRTR2S1PR1
SCHEMBL3281863 0.83 HCRTR1 (0.48) TNFHCRTR1HCRTR2CCR5
SCHEMBL4694248 0.83 ALDH1A1 (0.39) TNFALDH1A1HCRTR1HCRTR2S1PR1
SCHEMBL4695972 0.83 CHRNB2 (0.40) TNFALDH1A1HCRTR1HCRTR2KMT2A
SCHEMBL4692886 0.83 ALDH1A1 (0.42) TNFALDH1A1HCRTR1HCRTR2MEN1
SCHEMBL4695935 0.83 HCRTR2 (0.47) TNFALDH1A1HCRTR1HCRTR2
SCHEMBL4691604 0.83 GFER (0.42) TNFHCRTR1HCRTR2CHRM2MEN1
SCHEMBL4692864 0.82 TNF (0.35) TNFALDH1A1HCRTR1HCRTR2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed