SCHEMBL4692209

SCHEMBL4692209

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)C4CCCO4)CC3C2)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.46
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
MAPK1 P28482 1/20 0.41
POLB P06746 2/20 0.40
ALDH1A1 P00352 3/20 0.39
LMNA P02545 2/20 0.39
CYP3A4 P08684 1/20 0.38
PKM P14618 2/20 0.38
HPGD P15428 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5234052 0.83 PKM (0.46) KMT2ATSHRSMN1; SMN2MAPK1POLB
SCHEMBL4692183 0.83 TNF (0.35) ALDH1A1
SCHEMBL4695192 0.82 TNF (0.38) KMT2ASMN1; SMN2ALDH1A1PKMHPGD
SCHEMBL4691021 0.79 TNF (0.38) LMNA
SCHEMBL4690403 0.78 HCRTR1 (0.39) ALDH1A1HPGD
SCHEMBL3281863 0.78 HCRTR1 (0.48) KCNH2
SCHEMBL4694334 0.78 HCRTR1 (0.43)
SCHEMBL4695314 0.78 HCRTR1 (0.35) TSHRPOLBALDH1A1LMNAHPGD
SCHEMBL4692725 0.78 CHRNA4 (0.47) KMT2AALDH1A1HPGD
SCHEMBL4693718 0.78 TSHR (0.38) TSHRSMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed