SCHEMBL4695192

SCHEMBL4695192

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)C4C(C)(C)C4(C)C)CC3C2)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 2/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
TACR1 P25103 1/20 0.33
S1PR1 P21453 1/20 0.32
MGLL Q99685 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
SLC6A3 Q01959 2/20 0.31
PKM P14618 1/20 0.31
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30
ALDH1A1 P00352 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692886 0.83 ALDH1A1 (0.42) TNFMEN1KMT2AMGLLHCRTR1
SCHEMBL4691021 0.83 TNF (0.38) TNFTACR1S1PR1HCRTR1HCRTR2
SCHEMBL4692183 0.83 TNF (0.35) TNFTACR1SLC6A2SLC6A4SLC6A3
SCHEMBL4694334 0.82 HCRTR1 (0.43) TNFTACR1HCRTR1HCRTR2
SCHEMBL4690403 0.82 HCRTR1 (0.39) TNFTACR1S1PR1HCRTR1HCRTR2
SCHEMBL3281863 0.82 HCRTR1 (0.48) TNFHCRTR1HCRTR2
SCHEMBL4692209 0.82 KMT2A (0.46) KMT2APKMALDH1A1SMN1; SMN2HPGD
SCHEMBL4694354 0.82 P2RX7 (0.44) TNFHCRTR1HCRTR2
SCHEMBL4691868 0.82 HCRTR1 (0.47) TNFKMT2AHCRTR1HCRTR2ALDH1A1
SCHEMBL4695972 0.81 CHRNB2 (0.40) TNFKMT2AHCRTR1HCRTR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed