SCHEMBL4692183

SCHEMBL4692183

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)C4CCCCC4C)CC3C2)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.35
CNR2 P34972 4/20 0.34
ALDH1A1 P00352 2/20 0.34
CNR1 P21554 2/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
TACR1 P25103 1/20 0.33
GRM5 P41594 1/20 0.33
HTT P42858 1/20 0.33
CCR5 P51681 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
RAB9A P51151 1/20 0.32
SLC6A3 Q01959 3/20 0.31
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695192 0.83 TNF (0.38) TNFCNR2ALDH1A1CNR1PDE4A
SCHEMBL4692209 0.83 KMT2A (0.46) ALDH1A1
SCHEMBL4691021 0.80 TNF (0.38) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL4690403 0.79 HCRTR1 (0.39) TNFALDH1A1PDE4BTACR1CCR5
SCHEMBL4694334 0.79 HCRTR1 (0.43) TNFTACR1CCR5
SCHEMBL3281863 0.79 HCRTR1 (0.48) TNFCCR5
SCHEMBL4694815 0.79 HCRTR1 (0.37) TNFPDE4BCCR5
SCHEMBL4692886 0.78 ALDH1A1 (0.42) TNFALDH1A1HTTCCR5
SCHEMBL4695972 0.78 CHRNB2 (0.40) TNFALDH1A1
SCHEMBL4695935 0.78 HCRTR2 (0.47) TNFALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed