SCHEMBL5234052

SCHEMBL5234052

NC(=O)C[C@@H](c1ccccc1)N1CC2CN(C(=O)C3CCCO3)CC2C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.46
ALDH1A1 P00352 6/20 0.44
FASN P49327 2/20 0.43
TDP1 Q9NUW8 2/20 0.42
HPGD P15428 2/20 0.41
GAA P10253 2/20 0.41
KDM4E B2RXH2 3/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
TSHR P16473 2/20 0.38
HSD17B10 Q99714 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692209 0.83 KMT2A (0.46) PKMALDH1A1HPGDKMT2ASMN1; SMN2
SCHEMBL5229817 0.81 CCR5 (0.42) ALDH1A1TDP1
SCHEMBL5235854 0.79 PARP1 (0.37) TDP1HPGDCYP1A2CYP2C9MAPK1
SCHEMBL4689612 0.77 PKM (0.49) PKMALDH1A1FASNTDP1HPGD
SCHEMBL5237872 0.76 CCL5 (0.40) ALDH1A1TDP1HPGDKMT2AMEN1
SCHEMBL5233398 0.73 KDM4E (0.44) ALDH1A1TDP1HPGDGAAKDM4E
SCHEMBL5232470 0.73 CCR5 (0.54)
SCHEMBL5235643 0.72 CHRNB2 (0.53) ALDH1A1HPGDKDM4EHTTKMT2A
SCHEMBL5239176 0.72 HTT (0.43) PKMALDH1A1TDP1HPGDGAA
SCHEMBL5240008 0.72 ALDH1A1 (0.48) ALDH1A1GAAKDM4EHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed