SCHEMBL4692840

SCHEMBL4692840

NC(=O)c1ccccc1[CH]CCN1CC2CN(S(=O)(=O)c3ccccc3)C[C@@H]2C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
TGM2 P21980 2/20 0.39
F13A1 P00488 1/20 0.39
TGM1 P22735 1/20 0.39
ALDH1A1 P00352 3/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
KDM4E B2RXH2 1/20 0.36
PKM P14618 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
DRD2 P14416 1/20 0.36
HTR6 P50406 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694985 0.85 GRIN2B (0.44) PARP1GAADRD2
SCHEMBL3282844 0.85 GRIN2B (0.44) PARP1GAADRD2
SCHEMBL4694455 0.83 CHRNB2 (0.44) ALDH1A1KMT2ACHRNB2CHRNB4CHRNA3
SCHEMBL3284078 0.82 CHRNA4 (0.39) PARP1PARP2KDM4ECHRNB2CHRNB4
SCHEMBL4693059 0.81 CCR5 (0.37) PARP1ALDH1A1KMT2AKDM4ECHRNB2
SCHEMBL4691474 0.80 KDM4E (0.33) PARP1ALDH1A1KMT2AKDM4E
SCHEMBL4689903 0.79 P2RX7 (0.41) ALDH1A1GAAKMT2APOLB
SCHEMBL4693208 0.79 CCR5 (0.42) PARP1
SCHEMBL4692078 0.79 CCR5 (0.40) PARP1
SCHEMBL4691535 0.78 CCR5 (0.41) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed