SCHEMBL4693208

SCHEMBL4693208

NC(=O)c1ccccc1[CH]CCN1CC2CN(C(=O)C3CCCC3)C[C@@H]2C1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 7/20 0.42
CCL5 P13501 1/20 0.42
KCNK3 O14649 5/20 0.39
KCNK9 Q9NPC2 5/20 0.39
HSD11B1 P28845 1/20 0.39
PARP1 P09874 5/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691535 0.99 CCR5 (0.41) CCR5CCL5KCNK3KCNK9HSD11B1
SCHEMBL4692078 0.98 CCR5 (0.40) CCR5CCL5KCNK3KCNK9HSD11B1
SCHEMBL4693059 0.96 CCR5 (0.37) CCR5CCL5KCNK3KCNK9PARP1
SCHEMBL4691060 0.85 CCR5 (0.41) CCR5PARP1
SCHEMBL4696144 0.84 CCR5 (0.41) CCR5PARP1
SCHEMBL4689903 0.83 P2RX7 (0.41) CCR5
SCHEMBL4694455 0.82 CHRNB2 (0.44) CCR5
SCHEMBL4691474 0.81 KDM4E (0.33) CCR5PARP1
SCHEMBL4691802 0.81 CCR5 (0.48) CCR5
SCHEMBL4694234 0.81 ALDH1A1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed