SCHEMBL4694985

SCHEMBL4694985

NC(=O)c1ccccc1[CH]CCN1CC2CN(Cc3ccccc3)C[C@@H]2C1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 4/20 0.44
S1PR5 Q9H228 2/20 0.41
S1PR1 P21453 1/20 0.41
FUCA1 P04066 2/20 0.40
ADRA1D P25100 1/20 0.40
PARP1 P09874 2/20 0.39
GAA P10253 1/20 0.39
KCNH2 Q12809 1/20 0.38
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3282844 1.00 GRIN2B (0.44) GRIN2BS1PR5S1PR1FUCA1ADRA1D
SCHEMBL4694380 0.88 FAAH (0.41) S1PR5S1PR1KCNH2DRD2
SCHEMBL4692840 0.85 PARP1 (0.40) PARP1GAADRD2
SCHEMBL4690443 0.84 GRIN2B (0.37) GRIN2BDRD2DRD3
SCHEMBL4694455 0.84 CHRNB2 (0.44) KCNH2
SCHEMBL3284078 0.83 CHRNA4 (0.39) PARP1HRH3
SCHEMBL4694234 0.82 ALDH1A1 (0.41)
SCHEMBL4689903 0.82 P2RX7 (0.41) GAA
SCHEMBL4693659 0.82 CHRNB2 (0.47) GAA
SCHEMBL4693059 0.81 CCR5 (0.37) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed