SCHEMBL4696144

SCHEMBL4696144

NC(=O)c1ccccc1[CH]CCN1CC2CN(C(=O)CC3CCCCC3)C[C@@H]2C1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.41
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PARP1 P09874 3/20 0.35
BTK Q06187 1/20 0.33
SIRT2 Q8IXJ6 1/20 0.32
EPHX2 P34913 1/20 0.32
NAMPT P43490 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691060 0.99 CCR5 (0.41) CCR5KDM4EALDH1A1HSD17B10PARP1
SCHEMBL4691535 0.85 CCR5 (0.41) CCR5PARP1
SCHEMBL4693208 0.84 CCR5 (0.42) CCR5PARP1
SCHEMBL4691474 0.83 KDM4E (0.33) CCR5KDM4EALDH1A1PARP1
SCHEMBL4692078 0.82 CCR5 (0.40) CCR5PARP1
SCHEMBL4693059 0.82 CCR5 (0.37) CCR5KDM4EALDH1A1PARP1
SCHEMBL4694455 0.80 CHRNB2 (0.44) CCR5ALDH1A1
SCHEMBL4689903 0.78 P2RX7 (0.41) CCR5ALDH1A1
SCHEMBL3282844 0.77 GRIN2B (0.44) PARP1
SCHEMBL4694985 0.77 GRIN2B (0.44) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed