SCHEMBL4693291

SCHEMBL4693291

Cc1ccc(C(CC(N)=O)N2CC3CN(S(=O)(=O)c4cccs4)CC3C2)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
GAA P10253 2/20 0.44
PKM P14618 6/20 0.44
POLB P06746 1/20 0.42
RAB9A P51151 2/20 0.41
KMT2A Q03164 6/20 0.41
MEN1 O00255 5/20 0.41
NPC1 O15118 1/20 0.40
HTT P42858 1/20 0.40
APOBEC3A P31941 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692448 0.83 EPHX2 (0.46) ALDH1A1GAAKMT2AMEN1NPC1
SCHEMBL3283680 0.81 MAPT (0.41) ALDH1A1RAB9AHTT
SCHEMBL4695193 0.79 TRPV4 (0.40) PKMRAB9A
SCHEMBL4694340 0.79 TNF (0.36) ALDH1A1RAB9AKMT2AMEN1
SCHEMBL4695296 0.78 ALDH1A1 (0.48) ALDH1A1KMT2AMEN1HTT
SCHEMBL4694305 0.78 FPR2 (0.50) HTT
SCHEMBL3286926 0.78 TNF (0.41)
SCHEMBL4690881 0.77 SMN1; SMN2 (0.40) ALDH1A1PKMPOLBRAB9AKMT2A
SCHEMBL3281863 0.77 HCRTR1 (0.48)
SCHEMBL4696321 0.77 MAPT (0.40) RAB9AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed