SCHEMBL4692448

SCHEMBL4692448

Cc1cc(C)c(S(=O)(=O)N2CC3CN(C(CC(N)=O)c4ccc(C)c(Cl)c4)CC3C2)c(C)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 12/20 0.46
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
MAPK1 P28482 1/20 0.42
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
EBP Q15125 1/20 0.40
DHCR7 Q9UBM7 1/20 0.40
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694305 0.85 FPR2 (0.50) HTT
SCHEMBL4695296 0.85 ALDH1A1 (0.48) KMT2AMEN1MAPK1HTTALDH1A1
SCHEMBL4694334 0.84 HCRTR1 (0.43) EPHX2
SCHEMBL4693291 0.83 ALDH1A1 (0.44) KMT2AMEN1GAAHTTALDH1A1
SCHEMBL4690403 0.82 HCRTR1 (0.39) ALDH1A1
SCHEMBL4695193 0.82 TRPV4 (0.40) EPHX2MAPT
SCHEMBL3283680 0.82 MAPT (0.41) HTTALDH1A1MAPTNPSR1
SCHEMBL3286926 0.81 TNF (0.41) KDM4E
SCHEMBL4690738 0.80 HCRTR1 (0.46) HTTALDH1A1KDM4E
SCHEMBL4695935 0.79 HCRTR2 (0.47) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed