SCHEMBL4695296

SCHEMBL4695296

Cc1ccc(C(CC(N)=O)N2CC3CN(S(=O)(=O)c4c(C)noc4C)CC3C2)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
LMNA P02545 7/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
MAPT P10636 4/20 0.46
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
USP2 O75604 3/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 3/20 0.43
TSHR P16473 4/20 0.43
CHRM1 P11229 1/20 0.42
NPSR1 Q6W5P4 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692448 0.85 EPHX2 (0.46) ALDH1A1MAPTMEN1KMT2AMAPK1
SCHEMBL4694305 0.84 FPR2 (0.50) LMNASMN1; SMN2USP2HTTTSHR
SCHEMBL4691534 0.84 GFER (0.43) ALDH1A1LMNASMN1; SMN2MEN1KMT2A
SCHEMBL3283680 0.81 MAPT (0.41) ALDH1A1LMNASMN1; SMN2MAPTUSP2
SCHEMBL4693291 0.78 ALDH1A1 (0.44) ALDH1A1MEN1KMT2AHTT
SCHEMBL4695193 0.78 TRPV4 (0.40) MAPT
SCHEMBL4693944 0.77 CHRNA4 (0.41) ALDH1A1
SCHEMBL3286926 0.77 TNF (0.41) CHRM1
SCHEMBL4689556 0.76 LMNA (0.50) ALDH1A1LMNASMN1; SMN2KMT2AUSP2
SCHEMBL4690881 0.76 SMN1; SMN2 (0.40) ALDH1A1LMNASMN1; SMN2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed