SCHEMBL4693944

SCHEMBL4693944

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4cnoc4C)CC3C2)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNA4 P43681 1/20 0.41
HCRTR1 O43613 10/20 0.37
HCRTR2 O43614 10/20 0.37
TNF P01375 1/20 0.34
ACACB O00763 3/20 0.33
HRH4 Q9H3N8 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693625 0.85 HCRTR1 (0.37) HCRTR1HCRTR2TNFALDH1A1HPGD
SCHEMBL4691396 0.85 HCRTR1 (0.39) HCRTR1HCRTR2TNFCYP11B1CYP11B2
SCHEMBL4692886 0.84 ALDH1A1 (0.42) HCRTR1HCRTR2TNFALDH1A1HPGD
SCHEMBL4695935 0.84 HCRTR2 (0.47) HCRTR1HCRTR2TNFALDH1A1HPGD
SCHEMBL4691534 0.84 GFER (0.43) HCRTR1HCRTR2ALDH1A1
SCHEMBL4690680 0.83 HCRTR1 (0.42) HCRTR1HCRTR2TNFHRH4ALDH1A1
SCHEMBL4692692 0.83 HCRTR1 (0.45) HCRTR1HCRTR2TNFHRH4ALDH1A1
SCHEMBL4690738 0.83 HCRTR1 (0.46) HCRTR1HCRTR2TNFALDH1A1HPGD
SCHEMBL4693718 0.83 TSHR (0.38) HCRTR1HCRTR2TNFHPGD
SCHEMBL4694354 0.83 P2RX7 (0.44) HCRTR1HCRTR2TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed