SCHEMBL4690680

SCHEMBL4690680

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4ccc(Cl)cc4Cl)CC3C2)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.42
HCRTR2 O43614 4/20 0.42
P2RX7 Q99572 9/20 0.42
MAPT P10636 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
CHRM2 P08172 1/20 0.38
HRH4 Q9H3N8 1/20 0.37
TNF P01375 1/20 0.36
PDE2A O00408 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692692 0.92 HCRTR1 (0.45) HCRTR1HCRTR2MAPTALDH1A1HRH4
SCHEMBL4690738 0.89 HCRTR1 (0.46) HCRTR1HCRTR2P2RX7ALDH1A1HPGD
SCHEMBL4693625 0.88 HCRTR1 (0.37) HCRTR1HCRTR2P2RX7MAPTALDH1A1
SCHEMBL4694969 0.88 HCRTR1 (0.38) HCRTR1HCRTR2P2RX7HPGDHRH4
SCHEMBL4695935 0.87 HCRTR2 (0.47) HCRTR1HCRTR2P2RX7ALDH1A1HPGD
SCHEMBL4692886 0.87 ALDH1A1 (0.42) HCRTR1HCRTR2MAPTALDH1A1HPGD
SCHEMBL4694083 0.87 TSHR (0.40) HCRTR1HCRTR2MAPTALDH1A1HPGD
SCHEMBL4692712 0.86 HCRTR1 (0.43) HCRTR1HCRTR2P2RX7MAPTALDH1A1
SCHEMBL4694375 0.86 HCRTR1 (0.40) HCRTR1HCRTR2P2RX7MAPTALDH1A1
SCHEMBL4692944 0.86 HCRTR1 (0.41) HCRTR1HCRTR2P2RX7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed